Summary
AssigneeNeomorph
Filing years2022-2024
Patents2
Compounds95
Activity records195
Patent families2
Targets3
Assay familiesdegradation, selectivity
Activity metricsDC50, Dmax, IC50, degradation
Overview

Target distribution and active-compound trend

Target distribution

195 activity records

3 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

0316120222025
Activity compounds and values

Activity records

195 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C006076
% Degradation-=84%--IKZF2-MOLT-4CA3215907A1PGDB_A008119PGDB_C006076PGDB_AS002170View
2D structure for PGDB_C006093
DC50-=0.005uM-IKZF2-MOLT-4CA3215907A1PGDB_A008857PGDB_C006093PGDB_AS000536View
2D structure for PGDB_C006078
% Degradation-=81%--IKZF2-MOLT-4CA3215907A1PGDB_A010932PGDB_C006078PGDB_AS002170View
2D structure for PGDB_C006088
% Degradation-=79%--IKZF2-MOLT-4CA3215907A1PGDB_A011033PGDB_C006088PGDB_AS002170View
2D structure for PGDB_C006079
DC50-=0.006uM-IKZF2-MOLT-4CA3215907A1PGDB_A011307PGDB_C006079PGDB_AS000536View
2D structure for PGDB_C006095
% Degradation-=79%--IKZF2-MOLT-4CA3215907A1PGDB_A011698PGDB_C006095PGDB_AS002170View
2D structure for PGDB_C006083
% Degradation-=78%--IKZF2-MOLT-4CA3215907A1PGDB_A012761PGDB_C006083PGDB_AS002170View
2D structure for PGDB_C006105
% Degradation-=76%--IKZF2-MOLT-4CA3215907A1PGDB_A016883PGDB_C006105PGDB_AS002170View
2D structure for PGDB_C006077
% Degradation-=80%--IKZF2-MOLT-4CA3215907A1PGDB_A017114PGDB_C006077PGDB_AS002170View
2D structure for PGDB_C006097
DC50-=0.011uM-IKZF2-MOLT-4CA3215907A1PGDB_A018053PGDB_C006097PGDB_AS000536View
2D structure for PGDB_C006073
% Degradation-=90%--IKZF2-MOLT-4CA3215907A1PGDB_A021813PGDB_C006073PGDB_AS002170View
2D structure for PGDB_C006102
% Degradation-=69%--IKZF2-MOLT-4CA3215907A1PGDB_A022812PGDB_C006102PGDB_AS002170View
2D structure for PGDB_C006087
DC50-=0.021uM-IKZF2-MOLT-4CA3215907A1PGDB_A023963PGDB_C006087PGDB_AS000536View
2D structure for PGDB_C006081
DC50-=0.021uM-IKZF2-MOLT-4CA3215907A1PGDB_A027694PGDB_C006081PGDB_AS000536View
2D structure for PGDB_C006079
IC50-=23uM-KCNH2--CA3215907A1PGDB_A028498PGDB_C006079PGDB_AS002462View
2D structure for PGDB_C006085
DC50-=0.0083uM-IKZF2-MOLT-4CA3215907A1PGDB_A029615PGDB_C006085PGDB_AS000536View
2D structure for PGDB_C006095
DC50-=0.007uM-IKZF2-MOLT-4CA3215907A1PGDB_A030523PGDB_C006095PGDB_AS000536View
2D structure for PGDB_C006075
DC50-=0.031uM-IKZF2-MOLT-4CA3215907A1PGDB_A030619PGDB_C006075PGDB_AS000536View
2D structure for PGDB_C006092
DC50-=0.001uM-IKZF2-MOLT-4CA3215907A1PGDB_A031488PGDB_C006092PGDB_AS000536View
2D structure for PGDB_C006081
% Degradation-=71%--IKZF2-MOLT-4CA3215907A1PGDB_A031655PGDB_C006081PGDB_AS002170View