Summary
AssigneePeloton Therapeutics
Filing years2022
Patents1
Compounds100
Activity records279
Patent families1
Targets2
Assay familiesbinding, ternary_complex, viability
Activity metricsEC50, IC50
Overview

Target distribution and active-compound trend

Target distribution

279 activity records

2 targets

Active compounds by publication year

Distinct compounds linked to assignee patent publications

0501002024
Activity compounds and values

Activity records

279 records
Structure
Control
Value
ConcentrationTime
Record IDCompoundAssayDetails
2D structure for PGDB_C005605
EC50-=0.0026uM-RBM39DCAF15-AR127239A1PGDB_A008133PGDB_C005605PGDB_AS002536View
2D structure for PGDB_C005555
EC50-=0.0031uM-RBM39DCAF15-AR127239A1PGDB_A008138PGDB_C005555PGDB_AS002536View
2D structure for PGDB_C005569
IC50-=1.0678uM-DCAF15DCAF15-AR127239A1PGDB_A008577PGDB_C005569PGDB_AS000201View
2D structure for PGDB_C005599
EC50-=0.0011uM-RBM39DCAF15-AR127239A1PGDB_A008990PGDB_C005599PGDB_AS002536View
2D structure for PGDB_C005633
IC50-=1.791uM-RBM39-HCT116AR127239A1PGDB_A009052PGDB_C005633PGDB_AS002257View
2D structure for PGDB_C005627
EC50-=0.0007uM-RBM39DCAF15-AR127239A1PGDB_A009083PGDB_C005627PGDB_AS002536View
2D structure for PGDB_C005630
EC50-=0.0177uM-RBM39DCAF15-AR127239A1PGDB_A010054PGDB_C005630PGDB_AS002536View
2D structure for PGDB_C005554
IC50-=19.953uM-DCAF15DCAF15-AR127239A1PGDB_A010065PGDB_C005554PGDB_AS000201View
2D structure for PGDB_C005648
EC50-=0.2121uM-RBM39DCAF15-AR127239A1PGDB_A010317PGDB_C005648PGDB_AS002536View
2D structure for PGDB_C005583
IC50-=0.1257uM-RBM39-HCT116AR127239A1PGDB_A010379PGDB_C005583PGDB_AS002257View
2D structure for PGDB_C005574
IC50-=52.219uM-DCAF15DCAF15-AR127239A1PGDB_A010637PGDB_C005574PGDB_AS000201View
2D structure for PGDB_C005642
EC50-=0.0016uM-RBM39DCAF15-AR127239A1PGDB_A010891PGDB_C005642PGDB_AS002536View
2D structure for PGDB_C005557
IC50-=3.1602uM-RBM39-HCT116AR127239A1PGDB_A011726PGDB_C005557PGDB_AS002257View
2D structure for PGDB_C005612
IC50-=0.3513uM-RBM39-HCT116AR127239A1PGDB_A011735PGDB_C005612PGDB_AS002257View
2D structure for PGDB_C005584
EC50-=0.004uM-RBM39DCAF15-AR127239A1PGDB_A011874PGDB_C005584PGDB_AS002536View
2D structure for PGDB_C005570
IC50-=0.4146uM-RBM39-HCT116AR127239A1PGDB_A012296PGDB_C005570PGDB_AS002257View
2D structure for PGDB_C005559
IC50-=100uM-DCAF15DCAF15-AR127239A1PGDB_A012304PGDB_C005559PGDB_AS000201View
2D structure for PGDB_C005601
IC50-=0.5799uM-DCAF15DCAF15-AR127239A1PGDB_A012361PGDB_C005601PGDB_AS000201View
2D structure for PGDB_C005607
IC50-=5uM-RBM39-HCT116AR127239A1PGDB_A012439PGDB_C005607PGDB_AS002257View
2D structure for PGDB_C005640
IC50-=0.0518uM-DCAF15DCAF15-AR127239A1PGDB_A012701PGDB_C005640PGDB_AS000201View