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O=C1CC[C@H](N2Cc3cc(N4CCN(CC5CCN(c6ccc([C@@H]7c8ccc(O)cc8CC[C@@H]7c7ccccc7)cc6F)CC5)CC4)c4c(c3C2=O)OCO4)C(=O)N1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.9 | nM | - | — | ESR1 | - | MCF-7 | CN115611909A | PGDB_A011143 | PGDB_C006621 | PGDB_AS001650 | View | |
| IC50 | - | = | 0.5 | nM | - | — | ESR1 | - | - | CN115611909A | PGDB_A039560 | PGDB_C006621 | PGDB_AS002471 | View | |
| IC50 | - | = | 2.4 | nM | - | — | ESR1 | - | MCF-7 | CN115611909A | PGDB_A069913 | PGDB_C006621 | PGDB_AS000455 | View |