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Compound
PGDB_C026002
8 activity records1 related patents
2D structure
C[C@](O)(CNc1ccccc1-c1ccccc1)C(=O)Nc1ccc(C#N)c(C(F)(F)F)c1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| % Inhibition | - | = | 94 | % | 1 uM | - | - | - | - | JP2018513179A | PGDB_A012794 | PGDB_C026002 | PGDB_AS001050 | View |
| Emax | - | = | 18.6 | % | - | - | - | - | - | JP2018513179A | PGDB_A023047 | PGDB_C026002 | PGDB_AS000156 | View |
| Emax | - | = | 76.7 | % | - | - | - | - | - | JP2018513179A | PGDB_A025528 | PGDB_C026002 | PGDB_AS000006 | View |
| EC50 | - | = | 1.9 | nM | - | — | - | - | - | JP2018513179A | PGDB_A039168 | PGDB_C026002 | PGDB_AS000523 | View |
| % Inhibition | - | = | 63.8 | % | 1 uM | - | - | - | - | JP2018513179A | PGDB_A043229 | PGDB_C026002 | PGDB_AS000345 | View |
| IC50 | - | = | 305 | nM | - | — | - | - | - | JP2018513179A | PGDB_A047668 | PGDB_C026002 | PGDB_AS000864 | View |
| EC50 | - | > | 1000 | nM | - | — | - | - | - | JP2018513179A | PGDB_A053541 | PGDB_C026002 | PGDB_AS002549 | View |
| IC50 | - | = | 34.3 | nM | - | — | - | - | - | JP2018513179A | PGDB_A069669 | PGDB_C026002 | PGDB_AS000830 | View |