Loading compound
Loading detail record from the SQLite release...
Compound
PGDB_C028741
4 activity records1 related patents
2D structure
O=C1CCC(N2Cc3c(cc(N4CCN(c5ccc(OCc6ccccc6Cl)cc5)C(=O)C4)cc3C(F)F)C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| GI50 | - | = | 18.1 | nM | - | — | - | - | - | WO2026119815 | PGDB_A012064 | PGDB_C028741 | PGDB_AS000142 | View |
| Dmax | - | = | 93.3 | % | - | - | - | - | - | WO2026119815 | PGDB_A019681 | PGDB_C028741 | PGDB_AS002187 | View |
| % Inhibition | - | = | 85.4 | % | - | - | - | - | - | WO2026119815 | PGDB_A031815 | PGDB_C028741 | PGDB_AS001178 | View |
| DC50 | - | = | 8.1 | nM | - | — | - | - | - | WO2026119815 | PGDB_A054012 | PGDB_C028741 | PGDB_AS001959 | View |