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Compound
PGDB_C028855
4 activity records1 related patents
2D structure
O=C1CCC(N2Cc3ccc(N4CCN(c5cnc(Oc6ccccc6F)cn5)C(=O)C4)cc3C2=O)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| DC50 | - | = | 7.4 | nM | - | — | - | - | - | WO2026119815 | PGDB_A023478 | PGDB_C028855 | PGDB_AS001959 | View |
| % Inhibition | - | = | 94.8 | % | - | - | - | - | - | WO2026119815 | PGDB_A026971 | PGDB_C028855 | PGDB_AS001178 | View |
| Dmax | - | = | 82 | % | - | - | - | - | - | WO2026119815 | PGDB_A070405 | PGDB_C028855 | PGDB_AS002187 | View |
| GI50 | - | = | 137.6 | nM | - | — | - | - | - | WO2026119815 | PGDB_A071077 | PGDB_C028855 | PGDB_AS000142 | View |