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SIMM · NJU
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SIMM · NJU
Patent
EP4065576A1
70 compounds
105 activity records
2 assays
Patent summary
Publication number
EP4065576A1
Assignee
Captor Therapeutics
Family members
6
Family patent IDs
EP4065576A1
JP2023504143A
JP7760167B2
JPWO2021105335A5
US20230065745A1
WO2021105335A1
Filing year
2,020
Jurisdiction
EP
Compounds
70
Activity records
105
Assays
2
Activity compounds and values
Activity records
105 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
% Degradation
-
=
0-25
%
20 uM
24 h
-
-
NCI-H929
PGDB_A007529
PGDB_C025179
PGDB_AS001048
View
% Degradation
-
=
0-25
%
20 uM
24 h
-
-
NCI-H929
PGDB_A007601
PGDB_C025239
PGDB_AS001048
View
Ki
-
=
5-10
uM
-
—
-
-
-
PGDB_A007925
PGDB_C025206
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
PGDB_A008708
PGDB_C025177
PGDB_AS000901
View
Ki
-
>
10
uM
-
—
-
-
-
PGDB_A008803
PGDB_C025179
PGDB_AS000901
View
% Degradation
-
=
0-25
%
20 uM
24 h
-
-
NCI-H929
PGDB_A009120
PGDB_C025240
PGDB_AS001048
View
% Degradation
-
=
0-25
%
20 uM
24 h
-
-
NCI-H929
PGDB_A011386
PGDB_C025182
PGDB_AS001048
View
Ki
-
<
5
uM
-
—
-
-
-
PGDB_A012019
PGDB_C025196
PGDB_AS000901
View
Ki
-
>
10
uM
-
—
-
-
-
PGDB_A012243
PGDB_C025221
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
PGDB_A012313
PGDB_C025218
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
PGDB_A012622
PGDB_C025195
PGDB_AS000901
View
Ki
-
>
10
uM
-
—
-
-
-
PGDB_A012752
PGDB_C025189
PGDB_AS000901
View
% Degradation
-
=
0-25
%
20 uM
24 h
-
-
NCI-H929
PGDB_A014816
PGDB_C025236
PGDB_AS001048
View
Ki
-
<
5
uM
-
—
-
-
-
PGDB_A016428
PGDB_C025175
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
PGDB_A017147
PGDB_C025205
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
PGDB_A017864
PGDB_C025198
PGDB_AS000901
View
% Degradation
-
=
0-25
%
20 uM
24 h
-
-
NCI-H929
PGDB_A019073
PGDB_C025180
PGDB_AS001048
View
Ki
-
>
10
uM
-
—
-
-
-
PGDB_A019346
PGDB_C025201
PGDB_AS000901
View
Ki
-
=
5-10
uM
-
—
-
-
-
PGDB_A020118
PGDB_C025235
PGDB_AS000901
View
Ki
-
>
10
uM
-
—
-
-
-
PGDB_A022646
PGDB_C025204
PGDB_AS000901
View