PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Assay
PGDB_AS000901
System: biochemical
Target: CRBN
Assay context summary
Assay context
65 activity records
Assay family
binding
System
biochemical
Readout
Ki
Target
CRBN
E3
CRBN
Technology
fluorescence
Activity compounds and values
Activity records
65 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Ki
-
=
5-10
uM
-
—
-
-
-
EP4065576A1
PGDB_A007925
PGDB_C025206
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
EP4065576A1
PGDB_A008708
PGDB_C025177
PGDB_AS000901
View
Ki
-
>
10
uM
-
—
-
-
-
EP4065576A1
PGDB_A008803
PGDB_C025179
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
EP4065576A1
PGDB_A012019
PGDB_C025196
PGDB_AS000901
View
Ki
-
>
10
uM
-
—
-
-
-
EP4065576A1
PGDB_A012243
PGDB_C025221
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
EP4065576A1
PGDB_A012313
PGDB_C025218
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
EP4065576A1
PGDB_A012622
PGDB_C025195
PGDB_AS000901
View
Ki
-
>
10
uM
-
—
-
-
-
EP4065576A1
PGDB_A012752
PGDB_C025189
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
EP4065576A1
PGDB_A016428
PGDB_C025175
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
EP4065576A1
PGDB_A017147
PGDB_C025205
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
EP4065576A1
PGDB_A017864
PGDB_C025198
PGDB_AS000901
View
Ki
-
>
10
uM
-
—
-
-
-
EP4065576A1
PGDB_A019346
PGDB_C025201
PGDB_AS000901
View
Ki
-
=
5-10
uM
-
—
-
-
-
EP4065576A1
PGDB_A020118
PGDB_C025235
PGDB_AS000901
View
Ki
-
>
10
uM
-
—
-
-
-
EP4065576A1
PGDB_A022646
PGDB_C025204
PGDB_AS000901
View
Ki
-
>
10
uM
-
—
-
-
-
EP4065576A1
PGDB_A024240
PGDB_C025226
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
EP4065576A1
PGDB_A025469
PGDB_C025194
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
EP4065576A1
PGDB_A025787
PGDB_C025212
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
EP4065576A1
PGDB_A025819
PGDB_C025225
PGDB_AS000901
View
Ki
-
<
5
uM
-
—
-
-
-
EP4065576A1
PGDB_A026043
PGDB_C025199
PGDB_AS000901
View
Ki
-
>
10
uM
-
—
-
-
-
EP4065576A1
PGDB_A026754
PGDB_C025215
PGDB_AS000901
View