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SIMM · NJU
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SIMM · NJU
Patent
EP4540240A1
34 compounds
92 activity records
5 assays
Patent summary
Publication number
EP4540240A1
Assignee
Monte Rosa Therapeutics
Family members
3
Family patent IDs
EP4540240A1
US20250171420A1
WO2023244815A1
Filing year
2,023
Jurisdiction
EP
Compounds
34
Activity records
92
Assays
5
Activity compounds and values
Activity records
92 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
GI50
-
<=
0.1
uM
-
—
-
-
LS174T
PGDB_A007233
PGDB_C025247
PGDB_AS000256
View
GI50
-
>
0.1
uM
-
—
-
-
GP2D
PGDB_A008117
PGDB_C025253
PGDB_AS000507
View
GI50
-
<=
0.1
uM
-
—
-
-
GP2D
PGDB_A008246
PGDB_C025258
PGDB_AS000507
View
GI50
-
>
0.1
uM
-
—
-
-
LS180
PGDB_A009459
PGDB_C025257
PGDB_AS001295
View
GI50
-
<=
0.1
uM
-
—
-
-
GP2D
PGDB_A009627
PGDB_C025248
PGDB_AS000507
View
GI50
-
>
0.1
uM
-
—
-
-
GP2D
PGDB_A010447
PGDB_C025276
PGDB_AS000449
View
GI50
-
<=
0.1
uM
-
—
-
-
LS180
PGDB_A010843
PGDB_C010388
PGDB_AS001295
View
GI50
-
<=
0.1
uM
-
—
-
-
GP2D
PGDB_A011132
PGDB_C025259
PGDB_AS000507
View
GI50
-
>
0.1
uM
-
—
-
-
LS180
PGDB_A011489
PGDB_C025252
PGDB_AS001295
View
GI50
-
>
0.1
uM
-
—
-
-
LS174T
PGDB_A012005
PGDB_C025249
PGDB_AS000256
View
GI50
-
<=
0.1
uM
-
—
-
-
LS174T
PGDB_A015537
PGDB_C025265
PGDB_AS000256
View
GI50
-
<=
0.1
uM
-
—
-
-
LS174T
PGDB_A016756
PGDB_C025252
PGDB_AS000256
View
GI50
-
<=
0.1
uM
-
—
-
-
GP2D
PGDB_A020922
PGDB_C025245
PGDB_AS000507
View
GI50
-
<=
0.1
uM
-
—
-
-
GP2D
PGDB_A021478
PGDB_C025269
PGDB_AS000449
View
GI50
-
>
0.1
uM
-
—
-
-
LS174T
PGDB_A021549
PGDB_C025262
PGDB_AS000256
View
GI50
-
<=
0.1
uM
-
—
-
-
LS180
PGDB_A021639
PGDB_C025243
PGDB_AS001295
View
GI50
-
>
0.1
uM
-
—
-
-
GP2D
PGDB_A023026
PGDB_C025277
PGDB_AS001119
View
GI50
-
<=
0.1
uM
-
—
-
-
GP2D
PGDB_A026033
PGDB_C025277
PGDB_AS000449
View
GI50
-
>
0.1
uM
-
—
-
-
GP2D
PGDB_A026306
PGDB_C025272
PGDB_AS000449
View
GI50
-
>
0.1
uM
-
—
-
-
GP2D
PGDB_A026391
PGDB_C025276
PGDB_AS001119
View