Activity record

PGDB_A000668

Assay: viabilityTarget: VAV1QC: ambiguous
Activity overview

IC50 < 0.1 nM

TargetVAV1
Cell linepan-B
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS001700
PatentWO2026051943A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C029516
Compound IDPGDB_C029516
Compound实施例157
Source record IDPGDB_C029516
InChIKeyXEGRMHMTZVKOBU-UCFFOFKASA-N

Assay context

Assay IDPGDB_AS001700
Assay familyviability
Assay systemcell_based
ReadoutIC50
TargetVAV1
E3Not specified
Cell linepan-B
OrganismHomo sapiens

Source evidence

Patent IDWO2026051943A1
Compound location

实施例157

实施例157 enlarged structure实施例157 location on patent page 162
Activity table
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