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Compound
PGDB_C029516
5 activity records1 related patents
2D structure
CO[C@H]1CCN(C(=O)Nc2ccc(-c3cccc(C4CCC(=O)NC4=O)c3Cl)cc2C)C1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 0.1 | nM | - | — | VAV1 | - | pan-B | WO2026051943A1 | PGDB_A000668 | PGDB_C029516 | PGDB_AS001700 | View |
| IC50 | - | = | 0.1164 | nM | - | — | VAV1 | - | pan-B | WO2026051943A1 | PGDB_A001321 | PGDB_C029516 | PGDB_AS001016 | View |
| Dmax | - | = | 98.76 | % | Concentration series: 10 uM, 1 uM | - | VAV1 | - | - | WO2026051943A1 | PGDB_A003430 | PGDB_C029516 | PGDB_AS000777 | View |
| IC50 | - | = | 0.039 | nM | - | — | VAV1 | - | pan-T | WO2026051943A1 | PGDB_A005207 | PGDB_C029516 | PGDB_AS000112 | View |
| DC50 | - | = | 0.79 | nM | - | — | VAV1 | - | - | WO2026051943A1 | PGDB_A006162 | PGDB_C029516 | PGDB_AS001440 | View |