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SIMM · NJU

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A patent-derived molecular glue bioactivity database with traceable evidence.

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SIMM · NJU

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SIMM · NJU

Activity record

PGDB_A002472

Assay: % DegradationTarget: CSNK1A1QC: ambiguous

Activity overview

DC50 > 3000 nM

TargetCSNK1A1

E3 ligaseCRBN

Cell lineHEK293

Time18 h

Assay / Readoutluminescence / DC50

Assay IDPGDB_AS001709

PatentWO2026114958A1

QC statusambiguous

Evidence details

Compound, assay context, and source

Compound

Compound IDPGDB_C031990

CompoundI-51;I-51

Source record IDPGDB_C031990

InChIKeyGRCPZDFYZWKACH-BSSMAJELSA-N

Assay context

Assay IDPGDB_AS001709

Assay family% Degradation

Assay systemcell_based

ReadoutDC50

Technologyluminescence

Treatment time18 h

TargetCSNK1A1

E3CRBN

Cell lineHEK293

OrganismHomo sapiens

Source evidence

Patent IDWO2026114958A1

Compound location

I-51;I-51

I-51;I-51 enlarged structure

I-51;I-51 location on patent page 283

Activity table

Page 303 · table start

Page 304 · table middle

Page 305 · table end

A patent-derived molecular glue bioactivity database with traceable evidence.

Global reach

0

0 countries/regions

·

SIMM · NJU