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SIMM · NJU
Assay
PGDB_AS001709
System: cell_based
Target: CSNK1A1
Cell line: HEK293
Assay context summary
Assay context
58 activity records
Assay family
% Degradation
System
cell_based
Readout
DC50
Target
CSNK1A1
E3
Not specified
Cell line
HEK293
Organism
Homo sapiens
Technology
luminescence
Activity compounds and values
Activity records
58 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A000213
PGDB_C031956
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A000648
PGDB_C031959
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A000784
PGDB_C031976
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A000793
PGDB_C031972
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A000825
PGDB_C031945
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A001768
PGDB_C031997
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A001981
PGDB_C031977
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A002008
PGDB_C031976
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A002084
PGDB_C031951
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A002205
PGDB_C031979
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A002288
PGDB_C031963
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A002472
PGDB_C031990
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A002542
PGDB_C031960
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A002593
PGDB_C031965
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A002821
PGDB_C031971
PGDB_AS001709
View
DC50
-
=
53
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A002956
PGDB_C031986
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A003253
PGDB_C031942
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A003424
PGDB_C031947
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A003752
PGDB_C031946
PGDB_AS001709
View
DC50
-
>
3000
nM
-
—
CSNK1A1
CRBN
HEK293
WO2026114958A1
PGDB_A003830
PGDB_C031975
PGDB_AS001709
View