Activity record

PGDB_A003868

Assay: viabilityTarget: ARQC: standardized
Activity overview

IC50 = 0.006 nM

TargetAR
Cell lineVCaP
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS000271
PatentWO2026061104A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C029774
Compound IDPGDB_C029774
CompoundAR-P-249
Source record IDPGDB_C029774
InChIKeyJZGZWYTUBKNDJI-ZEVWKRCLSA-N

Assay context

Assay IDPGDB_AS000271
Assay familyviability
Assay systemcell_based
ReadoutIC50
Detection target% Cell viability
TargetAR
E3Not specified
Cell lineVCaP
OrganismHomo sapiens

Source evidence

Patent IDWO2026061104A1
Compound location

AR-P-249

AR-P-249 enlarged structureAR-P-249 location on patent page 189
Activity table
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