Activity record

PGDB_A004240

Assay: viabilityTarget: ARQC: standardized
Activity overview

IC50 = 0.0065 nM

TargetAR
Cell lineVCaP
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS000271
PatentWO2026061104A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C030004
Compound IDPGDB_C030004
CompoundAR-P-148
Source record IDPGDB_C029981
InChIKeyIPDABRXAUMIKLF-ARPOTICCSA-N

Assay context

Assay IDPGDB_AS000271
Assay familyviability
Assay systemcell_based
ReadoutIC50
Detection target% Cell viability
TargetAR
E3Not specified
Cell lineVCaP
OrganismHomo sapiens

Source evidence

Patent IDWO2026061104A1
Compound location

AR-P-148

AR-P-148 enlarged structureAR-P-148 location on patent page 155
Activity table
Page 272 · table start
Page 273 · table middle
Page 274 · table end