Activity record

PGDB_A005858

Assay: % DegradationTarget: CDK2QC: standardized
Activity overview

Dmax = 80.7 %

TargetCDK2
Cell lineHEK293T
Concentration10 uM
Assay / Readoutluminescence / Dmax
Assay IDPGDB_AS000752
PatentWO2026064643A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C030652
Compound IDPGDB_C030652
Compound3
Source record IDPGDB_C030652
InChIKeySXBALRQOQXWTIX-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000752
Assay family% Degradation
Assay systemcell_based
ReadoutDmax
Technologyluminescence
Concentration10 uM
TargetCDK2
E3Not specified
Cell lineHEK293T
OrganismHomo sapiens

Source evidence

Patent IDWO2026064643A1
Compound location

3

3 enlarged structure3 location on patent page 110
Activity table
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