Assay

PGDB_AS000752

System: cell_basedTarget: CDK2Cell line: HEK293T
Assay context summary

Assay context

10 activity records
Assay family% Degradation
Systemcell_based
ReadoutDmax
TargetCDK2
E3Not specified
Cell lineHEK293T
OrganismHomo sapiens
Technologyluminescence
Activity compounds and values

Activity records

10 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C030651
Dmax-=59.6%10 uM-CDK2-HEK293TWO2026064643A1PGDB_A004323PGDB_C030651PGDB_AS000752View
2D structure for PGDB_C011112
Dmax-=49.2%10 uM-CDK2-HEK293TWO2026064643A1PGDB_A004371PGDB_C011112PGDB_AS000752View
2D structure for PGDB_C026003
Dmax-=56.9%10 uM-CDK2-HEK293TWO2026064643A1PGDB_A004500PGDB_C026003PGDB_AS000752View
2D structure for PGDB_C030654
Dmax-=75.4%10 uM-CDK2-HEK293TWO2026064643A1PGDB_A005351PGDB_C030654PGDB_AS000752View
2D structure for PGDB_C030652
Dmax-=80.7%10 uM-CDK2-HEK293TWO2026064643A1PGDB_A005858PGDB_C030652PGDB_AS000752View
2D structure for PGDB_C025999
Dmax-=67%10 uM-CDK2-HEK293TWO2026064643A1PGDB_A078294PGDB_C025999PGDB_AS000752View
2D structure for PGDB_C011110
Dmax-=67.3%10 uM-CDK2-HEK293TWO2026064643A1PGDB_A079434PGDB_C011110PGDB_AS000752View
2D structure for PGDB_C030653
Dmax-=71.1%10 uM-CDK2-HEK293TWO2026064643A1PGDB_A079705PGDB_C030653PGDB_AS000752View
2D structure for PGDB_C030650
Dmax-=58.7%10 uM-CDK2-HEK293TWO2026064643A1PGDB_A080009PGDB_C030650PGDB_AS000752View
2D structure for PGDB_C026001
Dmax-=33%10 uM-CDK2-HEK293TWO2026064643A1PGDB_A080083PGDB_C026001PGDB_AS000752View
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