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SIMM · NJU
Activity record
PGDB_A006186
Assay: viability
Target: VAV1
QC: ambiguous
Activity overview
IC50 = 0.13 nM
Target
VAV1
Cell line
humanCD3T
Time
72 h
Assay / Readout
IC50 / viability
Assay ID
PGDB_AS000539
Patent
WO2026103873A1
QC status
ambiguous
Evidence details
Compound, assay context, and source
Compound
Compound ID
PGDB_C031405
Compound
69;69;化合物 69
Source record ID
PGDB_C031405
InChIKey
HQRGRANDPKIHIR-UHFFFAOYSA-N
Assay context
Assay ID
PGDB_AS000539
Assay family
viability
Assay system
cell_based
Readout
IC50
Treatment time
72 h
Target
VAV1
E3
Not specified
Cell line
humanCD3T
Organism
Homo sapiens
Source evidence
Patent ID
WO2026103873A1
Compound location
69;69;化合物 69
Activity table