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SIMM · NJU
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SIMM · NJU
Patent
WO2026103873A1
55 compounds
62 activity records
4 assays
Patent summary
Publication number
WO2026103873A1
Assignee
Hangzhou Baicreat Pharma-Tech Co Ltd
Title
HETEROCYCLIC COMPOUND AND PHARMACEUTICAL USE THEREOF
Family ID
unresolved_family_WO2026103873A1
Family members
1
Family patent IDs
WO2026103873A1
Filing year
2025
Publication date
2026-05-21
Jurisdiction
WO
Compounds
55
Activity records
62
Assays
4
Activity compounds and values
Activity records
62 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
DC50
-
=
45.09
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A000063
PGDB_C031440
PGDB_AS000831
View
DC50
-
=
13.11
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A000064
PGDB_C031456
PGDB_AS000831
View
DC50
-
=
9.04
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A000510
PGDB_C031416
PGDB_AS000831
View
IC50
-
=
0.14
nM
-
—
VAV1
-
humanCD3T
PGDB_A000561
PGDB_C031406
PGDB_AS000539
View
DC50
-
=
31.86
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A000709
PGDB_C029470
PGDB_AS000831
View
DC50
-
=
3.8
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A000756
PGDB_C031427
PGDB_AS000831
View
DC50
-
=
15.61
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A000933
PGDB_C031451
PGDB_AS000831
View
IC50
-
<
0.01
nM
-
—
VAV1
-
human CD3 T cells
PGDB_A001158
PGDB_C031404
PGDB_AS001232
View
DC50
-
=
1.69
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A001222
PGDB_C031415
PGDB_AS000831
View
DC50
-
=
11.57
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A001920
PGDB_C031413
PGDB_AS000831
View
DC50
-
=
15.82
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A001996
PGDB_C031417
PGDB_AS000831
View
DC50
-
=
26.47
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A002046
PGDB_C031445
PGDB_AS000831
View
DC50
-
=
5.86
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A002071
PGDB_C031446
PGDB_AS000831
View
DC50
-
=
3.43
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A002105
PGDB_C031421
PGDB_AS000831
View
DC50
-
=
11.82
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A002284
PGDB_C031434
PGDB_AS000831
View
DC50
-
=
30.62
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A002352
PGDB_C031437
PGDB_AS000831
View
DC50
-
=
9.71
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A002914
PGDB_C031438
PGDB_AS000831
View
DC50
-
=
6.67
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A003125
PGDB_C031431
PGDB_AS000831
View
DC50
-
=
37.26
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A003376
PGDB_C031448
PGDB_AS000831
View
DC50
-
=
15
nM
-
—
VAV1
-
293T-VAV1-FLAG
PGDB_A003426
PGDB_C031412
PGDB_AS000831
View
