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Compound
PGDB_C031405
4 activity records1 related patents
2D structure
O=C1CCC(c2cccc(-c3ccc(N4C(=O)c5ccnn5CC45CC5)cc3)c2Cl)C(=O)N1Compound summary
Physicochemical properties
Activity compounds and values
Activity records
| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 0.16 | nM | - | — | VAV1 | - | humanCD3T | WO2026103873A1 | PGDB_A004506 | PGDB_C031405 | PGDB_AS001038 | View |
| IC50 | - | = | 0.03 | nM | - | — | VAV1 | - | human CD3 T cells | WO2026103873A1 | PGDB_A005214 | PGDB_C031405 | PGDB_AS001232 | View |
| DC50 | - | = | 3.01 | nM | - | — | VAV1 | - | 293T-VAV1-FLAG | WO2026103873A1 | PGDB_A005383 | PGDB_C031405 | PGDB_AS000831 | View |
| IC50 | - | = | 0.13 | nM | - | — | VAV1 | - | humanCD3T | WO2026103873A1 | PGDB_A006186 | PGDB_C031405 | PGDB_AS000539 | View |