Activity record

PGDB_A007072

Assay: viabilityTarget: BTKQC: standardized
Activity overview

IC50 < 50 nM

TargetBTK
Cell lineMDA-MB-231
Time96 h
Assay / ReadoutCCK-8 / viability
Assay IDPGDB_AS001770
PatentCN116239566A
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C025809
Compound IDPGDB_C025809
CompoundGT-03287
Source record IDPGDB_C015979
InChIKeyWSIHFXFOAAVBFE-KSSJMHQNSA-N

Assay context

Assay IDPGDB_AS001770
Assay familyviability
Assay systemcell_based
Readoutviability
TechnologyCCK-8
Treatment time96 h
Detection target% Cell viability
TargetBTK
E3Not specified
Cell lineMDA-MB-231
OrganismHomo sapiens

Source evidence

Patent IDCN116239566A
Compound location

GT-03287

GT-03287 enlarged structureGT-03287 location on patent page 278
Activity table
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