Assay
PGDB_AS001770
System: cell_basedCell line: MDA-MB-231
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | < | 50 | nM | - | — | BTK | - | MDA-MB-231 | CN116239566A | PGDB_A007072 | PGDB_C025809 | PGDB_AS001770 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MDA-MB-231 | CN116239566A | PGDB_A010063 | PGDB_C025815 | PGDB_AS001770 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MDA-MB-231 | CN116239566A | PGDB_A022433 | PGDB_C019593 | PGDB_AS001770 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MDA-MB-231 | CN116239566A | PGDB_A026777 | PGDB_C015982 | PGDB_AS001770 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MDA-MB-231 | CN116239566A | PGDB_A034487 | PGDB_C025808 | PGDB_AS001770 | View | |
| IC50 | - | = | 100-500 | nM | - | — | BTK | - | MDA-MB-231 | CN116239566A | PGDB_A044342 | PGDB_C025803 | PGDB_AS001770 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MDA-MB-231 | CN116239566A | PGDB_A056639 | PGDB_C025807 | PGDB_AS001770 | View | |
| IC50 | - | = | 50-100 | nM | - | — | BTK | - | MDA-MB-231 | CN116239566A | PGDB_A062376 | PGDB_C025814 | PGDB_AS001770 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MDA-MB-231 | CN116239566A | PGDB_A066251 | PGDB_C025806 | PGDB_AS001770 | View | |
| IC50 | - | < | 50 | nM | - | — | BTK | - | MDA-MB-231 | CN116239566A | PGDB_A072849 | PGDB_C025813 | PGDB_AS001770 | View |