Activity record

PGDB_A007563

Assay: % DegradationTarget: ARQC: ambiguous
Activity overview

degradation = 48 %

TargetAR
Cell lineLNCaP
Concentration2.5 uM
Assay / Readout% Degradation
Assay IDPGDB_AS002020
PatentJP5998117B2
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C026007
Compound IDPGDB_C026007
CompoundASC-Q103
Source record IDPGDB_C026007
InChIKeyKOBSWMBBCVRSQI-UTLPMFLDSA-N

Assay context

Assay IDPGDB_AS002020
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration2.5 uM
Detection targetprotein_degradation
TargetAR
E3Not specified
Cell lineLNCaP
OrganismHomo sapiens

Source evidence

Patent IDJP5998117B2
Compound location

ASC-Q103

ASC-Q103 enlarged structureASC-Q103 location on patent page 61
Activity table
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