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SIMM · NJU
Assay
PGDB_AS002020
System: cell_based
Cell line: LNCaP
Assay context summary
Assay context
11 activity records
Assay family
% Degradation
System
cell_based
Readout
% Degradation
E3
Not specified
Cell line
LNCaP
Organism
Homo sapiens
Detection target
protein_degradation
Activity compounds and values
Activity records
11 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
% Degradation
-
=
48
%
2.5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A007563
PGDB_C026007
PGDB_AS002020
View
% Degradation
-
=
11
%
2.5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A011275
PGDB_C026013
PGDB_AS002020
View
% Degradation
-
=
0
%
2.5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A012620
PGDB_C026009
PGDB_AS002020
View
% Degradation
-
=
0
%
2.5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A020127
PGDB_C026016
PGDB_AS002020
View
% Degradation
-
=
15
%
2.5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A022076
PGDB_C026006
PGDB_AS002020
View
% Degradation
-
=
0
%
2.5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A055286
PGDB_C026010
PGDB_AS002020
View
% Degradation
-
=
21
%
2.5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A062099
PGDB_C026017
PGDB_AS002020
View
% Degradation
-
=
0
%
2.5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A067706
PGDB_C026011
PGDB_AS002020
View
% Degradation
-
=
4
%
2.5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A071401
PGDB_C026005
PGDB_AS002020
View
% Degradation
-
=
0
%
2.5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A073244
PGDB_C026014
PGDB_AS002020
View
% Degradation
-
=
22
%
2.5 uM
-
AR
-
LNCaP
JP5998117B2
PGDB_A073868
PGDB_C026015
PGDB_AS002020
View