Activity record

PGDB_A008240

Assay: ternary_complexTarget: RBM39QC: standardized
Activity overview

EC50 > 100 uM

TargetRBM39
E3 ligaseDCAF15
Time1 h
Assay / ReadoutAlphaLISA / EC50
Assay IDPGDB_AS000136
PatentWO2022173805A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C009647
Compound IDPGDB_C009647
Compound155
Source record IDPGDB_C009647
InChIKeyJEVSISFPCJTRRN-IBGZPJMESA-N

Assay context

Assay IDPGDB_AS000136
Assay familyternary_complex
Assay systembiochemical
ReadoutEC50
TechnologyAlphaLISA
Treatment time1 h
TargetRBM39
E3DCAF15

Source evidence

Patent IDWO2022173805A1
Compound location

155

155 enlarged structure155 location on patent page 148
Activity table
Page 171 · table start
Page 172 · table middle
Page 173 · table end