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SIMM · NJU
Assay
PGDB_AS000136
System: biochemical
Target: RBM39
Assay context summary
Assay context
174 activity records
Assay family
ternary_complex
System
biochemical
Readout
EC50
Target
RBM39
E3
DCAF15
Technology
AlphaLISA
Activity compounds and values
Activity records
174 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A007146
PGDB_C009790
PGDB_AS000136
View
EC50
-
>
100
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A008240
PGDB_C009647
PGDB_AS000136
View
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A008923
PGDB_C009677
PGDB_AS000136
View
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A009492
PGDB_C009646
PGDB_AS000136
View
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A010300
PGDB_C009654
PGDB_AS000136
View
EC50
-
<
100
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A011204
PGDB_C009735
PGDB_AS000136
View
EC50
-
<
1
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A011545
PGDB_C009624
PGDB_AS000136
View
EC50
-
<
1
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A012957
PGDB_C009728
PGDB_AS000136
View
EC50
-
>
100
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A013357
PGDB_C009736
PGDB_AS000136
View
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A013488
PGDB_C009684
PGDB_AS000136
View
EC50
-
<
1
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A013567
PGDB_C009717
PGDB_AS000136
View
EC50
-
<
1
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A013718
PGDB_C009627
PGDB_AS000136
View
EC50
-
<
1
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A013970
PGDB_C009701
PGDB_AS000136
View
EC50
-
<
1
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A014261
PGDB_C009752
PGDB_AS000136
View
EC50
-
>
100
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A015569
PGDB_C009741
PGDB_AS000136
View
EC50
-
<
1
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A015759
PGDB_C009666
PGDB_AS000136
View
EC50
-
<
1
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A015934
PGDB_C009729
PGDB_AS000136
View
EC50
-
<
10
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A016243
PGDB_C009758
PGDB_AS000136
View
EC50
-
>
100
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A017329
PGDB_C009710
PGDB_AS000136
View
EC50
-
>
100
uM
-
—
RBM39
DCAF15
-
WO2022173805A1
PGDB_A017598
PGDB_C009699
PGDB_AS000136
View