Activity record

PGDB_A008502

Assay: cellular_functionTarget: ESR1QC: ambiguous
Activity overview

IC50 = 5.2 nM

TargetESR1
Cell lineHEK293
Time20 h
Assay / Readoutfluorescence / IC50
Assay IDPGDB_AS000727
PatentCN115260206A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006617
Compound IDPGDB_C006617
Compound实施例7;实施例7
Source record IDPGDB_C006617
InChIKeyQCYSSVDCZIPQNW-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000727
Assay familycellular_function
Assay systemcell_based
ReadoutIC50
Technologyfluorescence
Treatment time20 h
TargetESR1
E3Not specified
Cell lineHEK293

Source evidence

Patent IDCN115260206A
Compound location

实施例7;实施例7

实施例7;实施例7 enlarged structure实施例7;实施例7 location on patent page 40
Activity table
Page 48 · table start