Assay
PGDB_AS000727
System: cell_basedCell line: HEK293
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
 | IC50 | - | = | 5.2 | nM | - | — | ESR1 | - | HEK293 | CN115260206A | PGDB_A008502 | PGDB_C006617 | PGDB_AS000727 | View |
 | IC50 | - | = | 10.1 | nM | - | — | ESR1 | - | HEK293 | CN115260206A | PGDB_A010851 | PGDB_C006615 | PGDB_AS000727 | View |
 | IC50 | - | = | 8.7 | nM | - | — | ESR1 | - | HEK293 | CN115260206A | PGDB_A014817 | PGDB_C006613 | PGDB_AS000727 | View |
 | IC50 | - | = | 14.5 | nM | - | — | ESR1 | - | HEK293 | CN115260206A | PGDB_A030709 | PGDB_C006620 | PGDB_AS000727 | View |
 | IC50 | - | = | 9.1 | nM | - | — | ESR1 | - | HEK293 | CN115260206A | PGDB_A039781 | PGDB_C006614 | PGDB_AS000727 | View |
 | IC50 | - | = | 4.9 | nM | - | — | ESR1 | - | HEK293 | CN115260206A | PGDB_A052245 | PGDB_C006618 | PGDB_AS000727 | View |
 | IC50 | - | = | 13.2 | nM | - | — | ESR1 | - | HEK293 | CN115260206A | PGDB_A065365 | PGDB_C006619 | PGDB_AS000727 | View |
 | IC50 | - | = | 7.3 | nM | - | — | ESR1 | - | HEK293 | CN115260206A | PGDB_A074912 | PGDB_C006616 | PGDB_AS000727 | View |