Activity record

PGDB_A008825

Assay: viabilityTarget: CDK12QC: ambiguous
Activity overview

IC50 = 1.6 nM

TargetCDK12
Cell lineA673
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS002570
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006594
Compound IDPGDB_C006594
CompoundH-APPAMP-027;H-APPAMP-027
Source record IDPGDB_C006594
InChIKeyRZTSBGXHEPIKKP-APWZRJJASA-N

Assay context

Assay IDPGDB_AS002570
Assay familyviability
Assay systemcell_based
ReadoutIC50
TargetCDK12
E3Not specified
Cell lineA673

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-027;H-APPAMP-027

H-APPAMP-027;H-APPAMP-027 enlarged structureH-APPAMP-027;H-APPAMP-027 location on patent page 43
Activity table
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