Assay

PGDB_AS002570

System: cell_basedTarget: CDK12Cell line: A673
Assay context summary

Assay context

45 activity records
Assay familyviability
Systemcell_based
ReadoutIC50
TargetCDK12
E3Not specified
Cell lineA673
Activity compounds and values

Activity records

45 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C006594
IC50-=1.6nM-—CDK12-A673CN114929708BPGDB_A008825PGDB_C006594PGDB_AS002570View
2D structure for PGDB_C006604
IC50-=18.1nM-—CDK12-A673CN114929708BPGDB_A011383PGDB_C006604PGDB_AS002570View
2D structure for PGDB_C006574
IC50-=27nM-—CDK12-A673CN114929708BPGDB_A012187PGDB_C006574PGDB_AS002570View
2D structure for PGDB_C006579
IC50-=21.8nM-—CDK12-A673CN114929708BPGDB_A013611PGDB_C006579PGDB_AS002570View
2D structure for PGDB_C006605
IC50-=4.6nM-—CDK12-A673CN114929708BPGDB_A013881PGDB_C006605PGDB_AS002570View
2D structure for PGDB_C006600
IC50-=5.7nM-—CDK12-A673CN114929708BPGDB_A020152PGDB_C006600PGDB_AS002570View
2D structure for PGDB_C006577
IC50-=4.3nM-—CDK12-A673CN114929708BPGDB_A021078PGDB_C006577PGDB_AS002570View
2D structure for PGDB_C006589
IC50-=10.3nM-—CDK12-A673CN114929708BPGDB_A021877PGDB_C006589PGDB_AS002570View
2D structure for PGDB_C006584
IC50-=8.3nM-—CDK12-A673CN114929708BPGDB_A022962PGDB_C006584PGDB_AS002570View
2D structure for PGDB_C006586
IC50-=76.9nM-—CDK12-A673CN114929708BPGDB_A024646PGDB_C006586PGDB_AS002570View
2D structure for PGDB_C006583
IC50-=14.8nM-—CDK12-A673CN114929708BPGDB_A029813PGDB_C006583PGDB_AS002570View
2D structure for PGDB_C006608
IC50-=9.8nM-—CDK12-A673CN114929708BPGDB_A030136PGDB_C006608PGDB_AS002570View
2D structure for PGDB_C006570
IC50-=8nM-—CDK12-A673CN114929708BPGDB_A032658PGDB_C006570PGDB_AS002570View
2D structure for PGDB_C006591
IC50-=19.8nM-—CDK12-A673CN114929708BPGDB_A033357PGDB_C006591PGDB_AS002570View
2D structure for PGDB_C006603
IC50-=10.4nM-—CDK12-A673CN114929708BPGDB_A033974PGDB_C006603PGDB_AS002570View
2D structure for PGDB_C006569
IC50-=716nM-—CDK12-A673CN114929708BPGDB_A037146PGDB_C006569PGDB_AS002570View
2D structure for PGDB_C006602
IC50-=17.3nM-—CDK12-A673CN114929708BPGDB_A039528PGDB_C006602PGDB_AS002570View
2D structure for PGDB_C006568
IC50-=123nM-—CDK12-A673CN114929708BPGDB_A039836PGDB_C006568PGDB_AS002570View
2D structure for PGDB_C006587
IC50-=115.5nM-—CDK12-A673CN114929708BPGDB_A041408PGDB_C006587PGDB_AS002570View
2D structure for PGDB_C006610
IC50-=340nM-—CDK12-A673CN114929708BPGDB_A043275PGDB_C006610PGDB_AS002570View
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