Activity record

PGDB_A010851

Assay: cellular_functionTarget: ESR1QC: ambiguous
Activity overview

IC50 = 10.1 nM

TargetESR1
Cell lineHEK293
Time20 h
Assay / Readoutfluorescence / IC50
Assay IDPGDB_AS000727
PatentCN115260206A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006615
Compound IDPGDB_C006615
Compound实施例3
Source record IDPGDB_C006615
InChIKeyYJIMOHYLHMYVGB-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000727
Assay familycellular_function
Assay systemcell_based
ReadoutIC50
Technologyfluorescence
Treatment time20 h
TargetESR1
E3Not specified
Cell lineHEK293

Source evidence

Patent IDCN115260206A
Compound location

实施例3

实施例3 enlarged structure实施例3 location on patent page 29
Activity table
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