Activity record

PGDB_A011897

Assay: % DegradationTarget: GSPT1QC: ambiguous
Activity overview

degradation = 9.7 %

TargetGSPT1
Concentration100 nM
Assay / Readout% Degradation
Assay IDPGDB_AS002431
PatentWO2024059107A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C002842
Compound IDPGDB_C002842
Compound91;91;91
Source record IDPGDB_C002842
InChIKeyNOGRJAPNDFXWLC-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002431
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration100 nM
Detection targetprotein_degradation
TargetGSPT1
E3Not specified

Source evidence

Patent IDWO2024059107A1
Compound location

91;91;91

91;91;91 enlarged structure91;91;91 location on patent page 12
Activity table
Page 141 · table single