Activity record

PGDB_A011916

Assay: bindingTarget: CRBNQC: standardized
Activity overview

Kd = 0.051 uM

TargetCRBN
E3 ligaseCRBN
Assay / ReadoutKd / binding
Assay IDPGDB_AS000522
PatentWO2025043225
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C008058
Compound IDPGDB_C008058
Compound128;128;128
Source record IDPGDB_C008058
InChIKeyFVOMAXBNUAFFMU-XYPWUTKMSA-N

Assay context

Assay IDPGDB_AS000522
Assay familybinding
Assay systembiochemical
ReadoutKd
TargetCRBN
E3CRBN

Source evidence

Patent IDWO2025043225
Compound location

128;128;128

128;128;128 enlarged structure128;128;128 location on patent page 42
Activity table
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