Assay

PGDB_AS000522

System: biochemicalTarget: CRBN
Assay context summary

Assay context

85 activity records
Assay familybinding
Systembiochemical
ReadoutKd
TargetCRBN
E3CRBN
Activity compounds and values

Activity records

85 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C008122
Kd-=0.13uM-—CRBNCRBN-WO2025043225PGDB_A007039PGDB_C008122PGDB_AS000522View
2D structure for PGDB_C008048
Kd-=0.017uM-—CRBNCRBN-WO2025043225PGDB_A008203PGDB_C008048PGDB_AS000522View
2D structure for PGDB_C008112
Kd-=0.047uM-—CRBNCRBN-WO2025043225PGDB_A008272PGDB_C008112PGDB_AS000522View
2D structure for PGDB_C008082
Kd-=1.3uM-—CRBNCRBN-WO2025043225PGDB_A009001PGDB_C008082PGDB_AS000522View
2D structure for PGDB_C008060
Kd-=0.065uM-—CRBNCRBN-WO2025043225PGDB_A009371PGDB_C008060PGDB_AS000522View
2D structure for PGDB_C008073
Kd-=0.015uM-—CRBNCRBN-WO2025043225PGDB_A010475PGDB_C008073PGDB_AS000522View
2D structure for PGDB_C008100
Kd-=0.33uM-—CRBNCRBN-WO2025043225PGDB_A011575PGDB_C008100PGDB_AS000522View
2D structure for PGDB_C008070
Kd-=0.0079uM-—CRBNCRBN-WO2025043225PGDB_A011757PGDB_C008070PGDB_AS000522View
2D structure for PGDB_C008055
Kd-=0.013uM-—CRBNCRBN-WO2025043225PGDB_A011792PGDB_C008055PGDB_AS000522View
2D structure for PGDB_C008058
Kd-=0.051uM-—CRBNCRBN-WO2025043225PGDB_A011916PGDB_C008058PGDB_AS000522View
2D structure for PGDB_C008110
Kd-=0.0051uM-—CRBNCRBN-WO2025043225PGDB_A012390PGDB_C008110PGDB_AS000522View
2D structure for PGDB_C008132
Kd-=0.16uM-—CRBNCRBN-WO2025043225PGDB_A012921PGDB_C008132PGDB_AS000522View
2D structure for PGDB_C008105
Kd-=0.14uM-—CRBNCRBN-WO2025043225PGDB_A013752PGDB_C008105PGDB_AS000522View
2D structure for PGDB_C008116
Kd-=0.15uM-—CRBNCRBN-WO2025043225PGDB_A014222PGDB_C008116PGDB_AS000522View
2D structure for PGDB_C008057
Kd-=0.031uM-—CRBNCRBN-WO2025043225PGDB_A014721PGDB_C008057PGDB_AS000522View
2D structure for PGDB_C008071
Kd-=0.088uM-—CRBNCRBN-WO2025043225PGDB_A015288PGDB_C008071PGDB_AS000522View
2D structure for PGDB_C008126
Kd-=0.7uM-—CRBNCRBN-WO2025043225PGDB_A016611PGDB_C008126PGDB_AS000522View
2D structure for PGDB_C008069
Kd-=0.0078uM-—CRBNCRBN-WO2025043225PGDB_A016785PGDB_C008069PGDB_AS000522View
2D structure for PGDB_C008065
Kd-=0.013uM-—CRBNCRBN-WO2025043225PGDB_A016787PGDB_C008065PGDB_AS000522View
2D structure for PGDB_C008072
Kd-=0.26uM-—CRBNCRBN-WO2025043225PGDB_A017557PGDB_C008072PGDB_AS000522View
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