Activity record

PGDB_A013684

Assay: biochemicalQC: ambiguous
Activity overview

selectivity_index = 0.1 fold

Time60 min
ControlCDK7 / CDK12
Assay / ReadoutFold change / biochemical
Assay IDPGDB_AS002236
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006590
Compound IDPGDB_C006590
CompoundH-APPAMP-023;H-APPAMP-023
Source record IDPGDB_C006590
InChIKeyOJMDASWRIMYSTE-QAPCUYQASA-N

Assay context

Assay IDPGDB_AS002236
Assay familybiochemical
Assay systembiochemical
ReadoutFold change
Treatment time60 min
TargetCDK12 | CDK7
E3Not specified
OrganismHomo sapiens

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-023;H-APPAMP-023

H-APPAMP-023;H-APPAMP-023 enlarged structureH-APPAMP-023;H-APPAMP-023 location on patent page 42
Activity table
Page 195 · table start
Page 196 · table middle
Page 197 · table end