Activity record

PGDB_A017124

Assay: % DegradationTarget: GSPT1QC: ambiguous
Activity overview

degradation = 12.2 %

TargetGSPT1
Concentration1 uM
Assay / Readout% Degradation
Assay IDPGDB_AS001974
PatentWO2024059107A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C002816
Compound IDPGDB_C002816
Compound52;52;52
Source record IDPGDB_C002816
InChIKeyUIFPBNRHYJGQSS-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001974
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration1 uM
Detection targetprotein_degradation
TargetGSPT1
E3Not specified

Source evidence

Patent IDWO2024059107A1
Compound location

52;52;52

52;52;52 enlarged structure52;52;52 location on patent page 9
Activity table
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