Assay

PGDB_AS001974

System: cell_basedTarget: GSPT1
Assay context summary

Assay context

44 activity records
Assay family% Degradation
Systemcell_based
Readout% Degradation
TargetGSPT1
E3Not specified
Detection targetprotein_degradation
Activity compounds and values

Activity records

44 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C002833
% Degradation-=44.3%1 uM-GSPT1--WO2024059107A1PGDB_A010722PGDB_C002833PGDB_AS001974View
2D structure for PGDB_C002832
% Degradation-=49%1 uM-GSPT1--WO2024059107A1PGDB_A015466PGDB_C002832PGDB_AS001974View
2D structure for PGDB_C002817
% Degradation-=1.2%1 uM-GSPT1--WO2024059107A1PGDB_A015763PGDB_C002817PGDB_AS001974View
2D structure for PGDB_C002816
% Degradation-=12.2%1 uM-GSPT1--WO2024059107A1PGDB_A017124PGDB_C002816PGDB_AS001974View
2D structure for PGDB_C002849
% Degradation-=6.2%1 uM-GSPT1--WO2024059107A1PGDB_A018807PGDB_C002849PGDB_AS001974View
2D structure for PGDB_C002822
% Degradation-=21.3%1 uM-GSPT1--WO2024059107A1PGDB_A018887PGDB_C002822PGDB_AS001974View
2D structure for PGDB_C002834
% Degradation-=14.4%1 uM-GSPT1--WO2024059107A1PGDB_A020203PGDB_C002834PGDB_AS001974View
2D structure for PGDB_C002811
% Degradation-=16.9%1 uM-GSPT1--WO2024059107A1PGDB_A021957PGDB_C002811PGDB_AS001974View
2D structure for PGDB_C002824
% Degradation-=16.5%1 uM-GSPT1--WO2024059107A1PGDB_A024816PGDB_C002824PGDB_AS001974View
2D structure for PGDB_C002829
% Degradation-=21.3%1 uM-GSPT1--WO2024059107A1PGDB_A025129PGDB_C002829PGDB_AS001974View
2D structure for PGDB_C002809
% Degradation-=11.1%1 uM-GSPT1--WO2024059107A1PGDB_A028785PGDB_C002809PGDB_AS001974View
2D structure for PGDB_C002847
% Degradation-=10.1%1 uM-GSPT1--WO2024059107A1PGDB_A029160PGDB_C002847PGDB_AS001974View
2D structure for PGDB_C002838
% Degradation-=11.9%1 uM-GSPT1--WO2024059107A1PGDB_A031506PGDB_C002838PGDB_AS001974View
2D structure for PGDB_C002842
% Degradation-=11.5%1 uM-GSPT1--WO2024059107A1PGDB_A034769PGDB_C002842PGDB_AS001974View
2D structure for PGDB_C002828
% Degradation-=12.6%1 uM-GSPT1--WO2024059107A1PGDB_A034864PGDB_C002828PGDB_AS001974View
2D structure for PGDB_C002815
% Degradation-=4%1 uM-GSPT1--WO2024059107A1PGDB_A038160PGDB_C002815PGDB_AS001974View
2D structure for PGDB_C002807
% Degradation-=8.6%1 uM-GSPT1--WO2024059107A1PGDB_A039803PGDB_C002807PGDB_AS001974View
2D structure for PGDB_C002823
% Degradation-=69.4%1 uM-GSPT1--WO2024059107A1PGDB_A040338PGDB_C002823PGDB_AS001974View
2D structure for PGDB_C002848
% Degradation-=-3.4%1 uM-GSPT1--WO2024059107A1PGDB_A042657PGDB_C002848PGDB_AS001974View
2D structure for PGDB_C002810
% Degradation-=14%1 uM-GSPT1--WO2024059107A1PGDB_A045189PGDB_C002810PGDB_AS001974View
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