Activity record

PGDB_A017459

Assay: % DegradationQC: ambiguous
Activity overview

Emax < 45 %

Concentration10 uM
Time<45%
Assay / Readoutluminescence / Emax
Assay IDPGDB_AS000576
PatentWO2022081927A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C016633
Compound IDPGDB_C016633
Compound61
Source record IDPGDB_C026762
InChIKeyAKUMKHBMOVVVIQ-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS000576
Assay family% Degradation
Assay systemcell_based
ReadoutEmax
Technologyluminescence
Concentration10 uM
Treatment time<45%
TargetGSPT1
E3Not specified
OrganismHomo sapiens

Source evidence

Patent IDWO2022081927A1
Compound location

61

61 enlarged structure61 location on patent page 527
Activity table
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Page 528 · table end