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CCOC(=O)c1ccc(Cc2ccc3c4c(cccc24)N(C2CCC(=O)NC2=O)C3=O)cc1| Structure | Control | Value | Concentration | Time | Record ID | Compound | Assay | Details | |||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| Emax | - | < | 45 | % | - | DC50 > 10000 nM | DC50 >= 100 nM and <= 1000 nM | DC50 < 100 nM | - | - | NCI-H929.11 | WO2022081927A1 | PGDB_A007170 | PGDB_C016633 | PGDB_AS001790 | View | |
| Emax | - | < | 45 | % | 10 uM | <45% | - | - | - | WO2022081927A1 | PGDB_A017459 | PGDB_C016633 | PGDB_AS000576 | View | |
| Emax | - | >= | 45 | % | - | DC50 > 10000 nM | > 100 nM | DC50 < 100 nM | - | - | 293T.114 | WO2022081927A1 | PGDB_A047765 | PGDB_C016633 | PGDB_AS000287 | View | |
| DC50 | - | < | 100 | nM | - | — | - | - | KELLY.2 | WO2022081927A1 | PGDB_A054029 | PGDB_C016633 | PGDB_AS001296 | View | |
| DC50 | - | > | 10000 | nM | - | — | - | - | 293T.114 | WO2022081927A1 | PGDB_A061026 | PGDB_C016633 | PGDB_AS001223 | View | |
| Emax | - | < | 45 | % | - | DC50 > 10000 nM | DC50 >= 100 nM and <= 1000 nM | > 100 nM | - | - | KELLY.2 | WO2022081927A1 | PGDB_A069892 | PGDB_C016633 | PGDB_AS000499 | View |