Activity record

PGDB_A018507

Assay: biochemicalQC: manual_curated
Activity overview

selectivity_index = 100-500 fold

Time120 min
ControlCDK1 / CDK12
Assay / Readoutselectivity_fold / biochemical
Assay IDPGDB_AS002417
PatentWO2025110815A1
QC statusmanual_curated
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C011002
Compound IDPGDB_C011002
Compound115
Source record IDPGDB_C011002
InChIKeyHKHCDZAAXKYDBN-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002417
Assay familybiochemical
Assay systembiochemical
Readoutselectivity_fold
Treatment time120 min
E3Not specified

Source evidence

Patent IDWO2025110815A1
Compound location

115

115 enlarged structure115 location on patent page 136
Activity table
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