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SIMM · NJU
Assay
PGDB_AS002417
System: biochemical
Assay context summary
Assay context
32 activity records
Assay family
biochemical
System
biochemical
Readout
selectivity_fold
E3
Not specified
Activity compounds and values
Activity records
32 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Patent
Record ID
Compound
Assay
Details
Selectivity index
CDK1 / CDK12
=
100-500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A007998
PGDB_C010952
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
>
500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A008572
PGDB_C010960
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
>
500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A008916
PGDB_C010920
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
=
100-500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A013838
PGDB_C010952
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
<=
100
fold
-
—
-
-
-
WO2025110815A1
PGDB_A014206
PGDB_C010917
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
>
500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A015839
PGDB_C010959
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
>
500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A016544
PGDB_C010925
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
=
100-500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A018507
PGDB_C011002
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
<=
100
fold
-
—
-
-
-
WO2025110815A1
PGDB_A019733
PGDB_C010951
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
<=
100
fold
-
—
-
-
-
WO2025110815A1
PGDB_A020733
PGDB_C010901
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
>
500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A023320
PGDB_C010958
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
=
100-500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A024844
PGDB_C010944
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
>
500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A025641
PGDB_C010958
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
=
100-500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A027741
PGDB_C011002
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
=
100-500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A032741
PGDB_C010954
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
>
500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A032873
PGDB_C010955
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
>
500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A033565
PGDB_C010960
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
>
500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A034821
PGDB_C010921
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
=
100-500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A039600
PGDB_C010944
PGDB_AS002417
View
Selectivity index
CDK1 / CDK12
>
500
fold
-
—
-
-
-
WO2025110815A1
PGDB_A046203
PGDB_C010955
PGDB_AS002417
View