Assay context summary

Assay context

32 activity records
Activity compounds and values

Activity records

32 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C010952
Selectivity indexCDK1 / CDK12=100-500fold----WO2025110815A1PGDB_A007998PGDB_C010952PGDB_AS002417View
2D structure for PGDB_C010960
Selectivity indexCDK1 / CDK12>500fold----WO2025110815A1PGDB_A008572PGDB_C010960PGDB_AS002417View
2D structure for PGDB_C010920
Selectivity indexCDK1 / CDK12>500fold----WO2025110815A1PGDB_A008916PGDB_C010920PGDB_AS002417View
2D structure for PGDB_C010952
Selectivity indexCDK1 / CDK12=100-500fold----WO2025110815A1PGDB_A013838PGDB_C010952PGDB_AS002417View
2D structure for PGDB_C010917
Selectivity indexCDK1 / CDK12<=100fold----WO2025110815A1PGDB_A014206PGDB_C010917PGDB_AS002417View
2D structure for PGDB_C010959
Selectivity indexCDK1 / CDK12>500fold----WO2025110815A1PGDB_A015839PGDB_C010959PGDB_AS002417View
2D structure for PGDB_C010925
Selectivity indexCDK1 / CDK12>500fold----WO2025110815A1PGDB_A016544PGDB_C010925PGDB_AS002417View
2D structure for PGDB_C011002
Selectivity indexCDK1 / CDK12=100-500fold----WO2025110815A1PGDB_A018507PGDB_C011002PGDB_AS002417View
2D structure for PGDB_C010951
Selectivity indexCDK1 / CDK12<=100fold----WO2025110815A1PGDB_A019733PGDB_C010951PGDB_AS002417View
2D structure for PGDB_C010901
Selectivity indexCDK1 / CDK12<=100fold----WO2025110815A1PGDB_A020733PGDB_C010901PGDB_AS002417View
2D structure for PGDB_C010958
Selectivity indexCDK1 / CDK12>500fold----WO2025110815A1PGDB_A023320PGDB_C010958PGDB_AS002417View
2D structure for PGDB_C010944
Selectivity indexCDK1 / CDK12=100-500fold----WO2025110815A1PGDB_A024844PGDB_C010944PGDB_AS002417View
2D structure for PGDB_C010958
Selectivity indexCDK1 / CDK12>500fold----WO2025110815A1PGDB_A025641PGDB_C010958PGDB_AS002417View
2D structure for PGDB_C011002
Selectivity indexCDK1 / CDK12=100-500fold----WO2025110815A1PGDB_A027741PGDB_C011002PGDB_AS002417View
2D structure for PGDB_C010954
Selectivity indexCDK1 / CDK12=100-500fold----WO2025110815A1PGDB_A032741PGDB_C010954PGDB_AS002417View
2D structure for PGDB_C010955
Selectivity indexCDK1 / CDK12>500fold----WO2025110815A1PGDB_A032873PGDB_C010955PGDB_AS002417View
2D structure for PGDB_C010960
Selectivity indexCDK1 / CDK12>500fold----WO2025110815A1PGDB_A033565PGDB_C010960PGDB_AS002417View
2D structure for PGDB_C010921
Selectivity indexCDK1 / CDK12>500fold----WO2025110815A1PGDB_A034821PGDB_C010921PGDB_AS002417View
2D structure for PGDB_C010944
Selectivity indexCDK1 / CDK12=100-500fold----WO2025110815A1PGDB_A039600PGDB_C010944PGDB_AS002417View
2D structure for PGDB_C010955
Selectivity indexCDK1 / CDK12>500fold----WO2025110815A1PGDB_A046203PGDB_C010955PGDB_AS002417View