Activity record

PGDB_A019080

Assay: % DegradationTarget: BRD4QC: ambiguous
Activity overview

degradation = 10-30 %

TargetBRD4
Concentration1 uM
Assay / ReadoutWestern_blot / % Degradation
Assay IDPGDB_AS002272
PatentCN117683022A
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C000059
Compound IDPGDB_C000059
CompoundCC-90009;CC-90009
Source record IDPGDB_C000059
InChIKeyPWBHUSLMHZLGRN-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS002272
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
TechnologyWestern_blot
Concentration1 uM
Detection targetprotein_degradation
TargetBRD4
E3Not specified

Source evidence

Patent IDCN117683022A
Compound location

CC-90009;CC-90009

CC-90009;CC-90009 enlarged structureCC-90009;CC-90009 location on patent page 5
Activity table
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