Assay

PGDB_AS002272

System: cell_basedTarget: BRD4
Assay context summary

Assay context

21 activity records
Assay family% Degradation
Systemcell_based
Readout% Degradation
TargetBRD4
E3Not specified
TechnologyWestern_blot
Detection targetprotein_degradation
Activity compounds and values

Activity records

21 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C000346
% Degradation-=30-60%1 uM-BRD4--CN117683022APGDB_A009721PGDB_C000346PGDB_AS002272View
2D structure for PGDB_C000354
% Degradation-=30-60%1 uM-BRD4--CN117683022APGDB_A016873PGDB_C000354PGDB_AS002272View
2D structure for PGDB_C000059
% Degradation-=10-30%1 uM-BRD4--CN117683022APGDB_A019080PGDB_C000059PGDB_AS002272View
2D structure for PGDB_C000353
% Degradation-=30-60%1 uM-BRD4--CN117683022APGDB_A021516PGDB_C000353PGDB_AS002272View
2D structure for PGDB_C000344
% Degradation-=10-30%1 uM-BRD4--CN117683022APGDB_A029149PGDB_C000344PGDB_AS002272View
2D structure for PGDB_C000355
% Degradation-=30-60%1 uM-BRD4--CN117683022APGDB_A032566PGDB_C000355PGDB_AS002272View
2D structure for PGDB_C000347
% Degradation-=30-60%1 uM-BRD4--CN117683022APGDB_A032731PGDB_C000347PGDB_AS002272View
2D structure for PGDB_C000341
% Degradation-=10-30%1 uM-BRD4--CN117683022APGDB_A032872PGDB_C000341PGDB_AS002272View
2D structure for PGDB_C000352
% Degradation-=10-30%1 uM-BRD4--CN117683022APGDB_A033245PGDB_C000352PGDB_AS002272View
2D structure for PGDB_C000339
% Degradation-=10-30%1 uM-BRD4--CN117683022APGDB_A041429PGDB_C000339PGDB_AS002272View
2D structure for PGDB_C000358
% Degradation-=30-60%1 uM-BRD4--CN117683022APGDB_A044553PGDB_C000358PGDB_AS002272View
2D structure for PGDB_C000345
% Degradation-=30-60%1 uM-BRD4--CN117683022APGDB_A044581PGDB_C000345PGDB_AS002272View
2D structure for PGDB_C000343
% Degradation-=10-30%1 uM-BRD4--CN117683022APGDB_A045684PGDB_C000343PGDB_AS002272View
2D structure for PGDB_C000357
% Degradation-=30-60%1 uM-BRD4--CN117683022APGDB_A047653PGDB_C000357PGDB_AS002272View
2D structure for PGDB_C000350
% Degradation-=30-60%1 uM-BRD4--CN117683022APGDB_A053352PGDB_C000350PGDB_AS002272View
2D structure for PGDB_C000340
% Degradation-=10-30%1 uM-BRD4--CN117683022APGDB_A060060PGDB_C000340PGDB_AS002272View
2D structure for PGDB_C000349
% Degradation-=30-60%1 uM-BRD4--CN117683022APGDB_A065438PGDB_C000349PGDB_AS002272View
2D structure for PGDB_C000342
% Degradation-=10-30%1 uM-BRD4--CN117683022APGDB_A068778PGDB_C000342PGDB_AS002272View
2D structure for PGDB_C000351
% Degradation-=10-30%1 uM-BRD4--CN117683022APGDB_A068817PGDB_C000351PGDB_AS002272View
2D structure for PGDB_C000348
% Degradation-=10-30%1 uM-BRD4--CN117683022APGDB_A075472PGDB_C000348PGDB_AS002272View
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