Activity record

PGDB_A020203

Assay: % DegradationTarget: GSPT1QC: ambiguous
Activity overview

degradation = 14.4 %

TargetGSPT1
Concentration1 uM
Assay / Readout% Degradation
Assay IDPGDB_AS001974
PatentWO2024059107A1
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C002834
Compound IDPGDB_C002834
Compound78;78;78
Source record IDPGDB_C002834
InChIKeyAOZLNZRSVIVLQX-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001974
Assay family% Degradation
Assay systemcell_based
Readout% Degradation
Concentration1 uM
Detection targetprotein_degradation
TargetGSPT1
E3Not specified

Source evidence

Patent IDWO2024059107A1
Compound location

78;78;78

78;78;78 enlarged structure78;78;78 location on patent page 11
Activity table
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