Activity record

PGDB_A021483

Assay: viabilityTarget: GSPT1QC: standardized
Activity overview

IC50 = 1.9 nM

TargetGSPT1
Cell lineMOLM-13
TimeThree days later
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS001795
PatentWO2022073469A1
QC statusstandardized
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C004674
Compound IDPGDB_C004674
CompoundGS-002;GS-002
Source record IDPGDB_C004674
InChIKeyIYUXBKRFBLWLOQ-UHFFFAOYSA-N

Assay context

Assay IDPGDB_AS001795
Assay familyviability
Assay systemcell_based
ReadoutIC50
Treatment timeThree days later
Detection target% Cell viability
TargetGSPT1
E3Not specified
Cell lineMOLM-13

Source evidence

Patent IDWO2022073469A1
Compound location

GS-002;GS-002

GS-002;GS-002 enlarged structureGS-002;GS-002 location on patent page 75
Activity table
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