Assay context summary

Assay context

26 activity records
Activity compounds and values

Activity records

26 records
StructureMetricControlRelationValueUnitConcentrationTimeTargetE3Cell linePatentRecord IDCompoundAssayDetails
2D structure for PGDB_C004678
IC50-=0.3nM-GSPT1-MOLM-13WO2022073469A1PGDB_A008983PGDB_C004678PGDB_AS001795View
2D structure for PGDB_C004679
IC50-=32nM-GSPT1-MOLM-13WO2022073469A1PGDB_A012298PGDB_C004679PGDB_AS001795View
2D structure for PGDB_C004691
IC50-=7nM-GSPT1-MOLM-13WO2022073469A1PGDB_A016274PGDB_C004691PGDB_AS001795View
2D structure for PGDB_C004697
IC50-=3680nM-GSPT1-MOLM-13WO2022073469A1PGDB_A019201PGDB_C004697PGDB_AS001795View
2D structure for PGDB_C004685
IC50-=1848nM-GSPT1-MOLM-13WO2022073469A1PGDB_A020818PGDB_C004685PGDB_AS001795View
2D structure for PGDB_C004674
IC50-=1.9nM-GSPT1-MOLM-13WO2022073469A1PGDB_A021483PGDB_C004674PGDB_AS001795View
2D structure for PGDB_C004695
IC50-=0.06nM-GSPT1-MOLM-13WO2022073469A1PGDB_A021744PGDB_C004695PGDB_AS001795View
2D structure for PGDB_C004673
IC50-=27nM-GSPT1-MOLM-13WO2022073469A1PGDB_A022731PGDB_C004673PGDB_AS001795View
2D structure for PGDB_C004677
IC50-=0.2nM-GSPT1-MOLM-13WO2022073469A1PGDB_A023922PGDB_C004677PGDB_AS001795View
2D structure for PGDB_C004680
IC50-=14nM-GSPT1-MOLM-13WO2022073469A1PGDB_A026064PGDB_C004680PGDB_AS001795View
2D structure for PGDB_C004696
IC50-=72nM-GSPT1-MOLM-13WO2022073469A1PGDB_A028500PGDB_C004696PGDB_AS001795View
2D structure for PGDB_C004684
IC50-=312nM-GSPT1-MOLM-13WO2022073469A1PGDB_A030796PGDB_C004684PGDB_AS001795View
2D structure for PGDB_C004698
IC50-=600nM-GSPT1-MOLM-13WO2022073469A1PGDB_A032021PGDB_C004698PGDB_AS001795View
2D structure for PGDB_C004676
IC50-=0.2nM-GSPT1-MOLM-13WO2022073469A1PGDB_A035820PGDB_C004676PGDB_AS001795View
2D structure for PGDB_C004682
IC50-=0.3nM-GSPT1-MOLM-13WO2022073469A1PGDB_A035929PGDB_C004682PGDB_AS001795View
2D structure for PGDB_C004681
IC50-=18nM-GSPT1-MOLM-13WO2022073469A1PGDB_A037320PGDB_C004681PGDB_AS001795View
2D structure for PGDB_C004687
IC50-=30nM-GSPT1-MOLM-13WO2022073469A1PGDB_A039688PGDB_C004687PGDB_AS001795View
2D structure for PGDB_C004688
IC50-=86nM-GSPT1-MOLM-13WO2022073469A1PGDB_A042875PGDB_C004688PGDB_AS001795View
2D structure for PGDB_C004686
IC50-=10nM-GSPT1-MOLM-13WO2022073469A1PGDB_A046946PGDB_C004686PGDB_AS001795View
2D structure for PGDB_C004694
IC50-=106nM-GSPT1-MOLM-13WO2022073469A1PGDB_A050878PGDB_C004694PGDB_AS001795View