PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Loading patent
Loading detail record from the SQLite release...
PatGlueDB
Search
Browse
Statistics
Contact
Help
·
SIMM · NJU
Patent
WO2022073469A1
621 compounds
2,503 activity records
8 assays
Patent summary
Publication number
WO2022073469A1
Assignee
Cullgen Shanghai
Title
Compounds and methods of treating cancers
Family ID
81125595
Family members
7
Family patent IDs
CN116583509A
EP4225749A1
EP4225749A4
JP2023545274A
US20240050428A1
US2024050428A1
WO2022073469A1
Filing year
2021
Publication date
2022-04-14
Jurisdiction
WO
Compounds
621
Activity records
2,503
Assays
8
Activity compounds and values
Activity records
2,503 records
Structure
Metric
Control
Relation
Value
Unit
Concentration
Time
Target
E3
Cell line
Record ID
Compound
Assay
Details
IC50
-
=
100-1000
nM
-
—
-
-
MV-4-11
PGDB_A007018
PGDB_C004856
PGDB_AS000609
View
IC50
-
=
100-1000
nM
-
—
GSPT1
-
MOLM-13
PGDB_A007038
PGDB_C005160
PGDB_AS000571
View
IC50
-
=
10-100
nM
-
—
-
-
MV-4-11
PGDB_A007046
PGDB_C004967
PGDB_AS002199
View
IC50
-
=
10-100
nM
-
—
-
-
MV-4-11
PGDB_A007075
PGDB_C005151
PGDB_AS002199
View
IC50
-
<
10
nM
-
—
GSPT1
-
MOLM-13
PGDB_A007079
PGDB_C004917
PGDB_AS000952
View
IC50
-
>=
1
uM
-
—
GSPT1
-
MOLM-13
PGDB_A007089
PGDB_C005286
PGDB_AS000571
View
IC50
-
=
10-100
nM
-
—
GSPT1
-
MOLM-13
PGDB_A007106
PGDB_C004920
PGDB_AS000571
View
IC50
-
>=
1
uM
-
—
GSPT1
-
MOLM-13
PGDB_A007114
PGDB_C004826
PGDB_AS000571
View
IC50
-
<
10
nM
-
—
GSPT1
-
MOLM-13
PGDB_A007213
PGDB_C005098
PGDB_AS000952
View
IC50
-
=
100-1000
nM
-
—
GSPT1
-
MOLM-13
PGDB_A007231
PGDB_C005187
PGDB_AS000952
View
IC50
-
=
100-1000
nM
-
—
-
-
MV-4-11
PGDB_A007235
PGDB_C004750
PGDB_AS000609
View
IC50
-
=
100-1000
nM
-
—
-
-
MV-4-11
PGDB_A007236
PGDB_C005157
PGDB_AS000609
View
IC50
-
>=
1
uM
-
—
GSPT1
-
MOLM-13
PGDB_A007259
PGDB_C004836
PGDB_AS000571
View
IC50
-
>=
1
uM
-
—
GSPT1
-
MOLM-13
PGDB_A007280
PGDB_C005134
PGDB_AS000571
View
IC50
-
>=
1
uM
-
—
-
-
MV-4-11
PGDB_A007285
PGDB_C004944
PGDB_AS000609
View
IC50
-
=
10-100
nM
-
—
-
-
MV-4-11
PGDB_A007406
PGDB_C004946
PGDB_AS002199
View
IC50
-
=
100-1000
nM
-
—
-
-
MV-4-11
PGDB_A007448
PGDB_C005049
PGDB_AS000609
View
IC50
-
>=
1
uM
-
—
GSPT1
-
MOLM-13
PGDB_A007462
PGDB_C004718
PGDB_AS000571
View
IC50
-
=
100-1000
nM
-
—
GSPT1
-
MOLM-13
PGDB_A007480
PGDB_C004985
PGDB_AS000571
View
IC50
-
>
10000
nM
-
—
-
-
MV-4-11
PGDB_A007520
PGDB_C004673
PGDB_AS001286
View