Activity record

PGDB_A022962

Assay: viabilityTarget: CDK12QC: ambiguous
Activity overview

IC50 = 8.3 nM

TargetCDK12
Cell lineA673
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS002570
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006584
Compound IDPGDB_C006584
CompoundH-APPAMP-017;H-APPAMP-017
Source record IDPGDB_C006584
InChIKeyCDFCOIXVUBLESU-XLIONFOSSA-N

Assay context

Assay IDPGDB_AS002570
Assay familyviability
Assay systemcell_based
ReadoutIC50
TargetCDK12
E3Not specified
Cell lineA673

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-017;H-APPAMP-017

H-APPAMP-017;H-APPAMP-017 enlarged structureH-APPAMP-017;H-APPAMP-017 location on patent page 40
Activity table
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