Activity record

PGDB_A024634

Assay: viabilityTarget: CDK12QC: ambiguous
Activity overview

IC50 = 44 nM

TargetCDK12
Cell lineA673
Assay / ReadoutIC50 / viability
Assay IDPGDB_AS002202
PatentCN114929708B
QC statusambiguous
Evidence details

Compound, assay context, and source

Compound

2D structure for PGDB_C006611
Compound IDPGDB_C006611
CompoundH-APPAMP-044
Source record IDPGDB_C006611
InChIKeyRXLOGDAYDFDLGX-QUCCMNQESA-N

Assay context

Assay IDPGDB_AS002202
Assay familyviability
Assay systemcell_based
ReadoutIC50
TargetCDK12 | CCNK
E3Not specified
Cell lineA673

Source evidence

Patent IDCN114929708B
Compound location

H-APPAMP-044

H-APPAMP-044 enlarged structureH-APPAMP-044 location on patent page 47
Activity table
Page 197 · table single