Assay
PGDB_AS002202
System: cell_basedTarget: CDK12 | CCNKCell line: A673
Assay context summary
Assay context
Activity compounds and values
Activity records
| Structure | Metric | Control | Relation | Value | Unit | Concentration | Time | Target | E3 | Cell line | Patent | Record ID | Compound | Assay | Details |
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
| IC50 | - | = | 110 | nM | - | — | CDK12 | - | A673 | CN114929708B | PGDB_A012469 | PGDB_C006612 | PGDB_AS002202 | View | |
| IC50 | - | = | 1.5 | nM | - | — | CDK12 | - | A673 | CN114929708B | PGDB_A019117 | PGDB_C006592 | PGDB_AS002202 | View | |
| IC50 | - | = | 44 | nM | - | — | CDK12 | - | A673 | CN114929708B | PGDB_A024634 | PGDB_C006611 | PGDB_AS002202 | View | |
| IC50 | - | = | 8.9 | nM | - | — | CDK12 | - | A673 | CN114929708B | PGDB_A029905 | PGDB_C006571 | PGDB_AS002202 | View | |
| IC50 | - | = | 340 | nM | - | — | CDK12 | - | A673 | CN114929708B | PGDB_A075544 | PGDB_C006610 | PGDB_AS002202 | View |